SCHEMBL5773536

SCHEMBL5773536

Fc1cc(Br)c2c(Sc3ccc(Cl)cc3)c3n(c2c1)CC[CH]3

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 14/20 0.56
PTGDR2 Q9Y5Y4 3/20 0.39
AKR1B1 P15121 2/20 0.34
PDE2A O00408 2/20 0.31
PTGDR Q13258 2/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777733 0.86 TBXA2R (0.42) TBXA2RPTGDR2HTR1ADRD2DRD4
SCHEMBL5778173 0.81 TBXA2R (0.50) TBXA2RPTGDR2AKR1B1PDE2APTGDR
SCHEMBL5776535 0.81 TBXA2R (0.39) TBXA2RPTGDR2
SCHEMBL5778034 0.79 TBXA2R (0.43) TBXA2RPDE2APTGDRHTR1ADRD2
SCHEMBL5773541 0.78 TBXA2R (0.55) TBXA2RPTGDR2AKR1B1PDE2APTGDR
SCHEMBL5779000 0.76 TBXA2R (0.55) TBXA2RPTGDR2AKR1B1PDE2APTGDR
SCHEMBL5777302 0.72 TBXA2R (0.33) TBXA2RPTGDR2AKR1B1HTR1A
SCHEMBL5773893 0.72 TBXA2R (1.00) TBXA2RPTGDR2PDE2APTGDR
SCHEMBL5774333 0.71 TBXA2R (0.67) TBXA2RPTGDR2PDE2APTGDR
SCHEMBL5837002 0.71 TBXA2R (0.71) TBXA2RPTGDR2PDE2APTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed