Brucine

Brucine

SCHEMBL577756

COc1cc2c(cc1OC)[C@@]13CCN4CC5=CCO[C@H]6CC(=O)N2[C@H]1[C@H]6[C@H]5C[C@H]43.OB(O)F.OB(O)F.OB(O)F.OB(O)F

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAS2R10 Q9NYW0 2/20 0.91
CHRM1 P11229 1/20 0.91
SMN1; SMN2 Q16637 1/20 0.91
GLRA1 P23415 14/20 0.67
GLRB P48167 14/20 0.67
CYP3A4 P08684 2/20 0.65
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
SCN1A P35498 1/20 0.65
TAS2R46 P59540 1/20 0.65
SCN2A Q99250 1/20 0.65
SCN3A Q9NY46 1/20 0.65
CYP1A2 P05177 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Brucine SCHEMBL31317695 0.96 TAS2R10 (0.98) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL7253414 0.96 TAS2R10 (0.98) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL10307298 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL113229 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL1648976 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL23468158 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL19476145 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL12293782 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL14029321 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL29391712 0.95 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418190-B1 The method of preparation of enantiomerically enriched products of condensation from racemic acids or acids of the low enentiomeric purity POLITECHNIKA LODZKA (PL) 2013-08-28 EP disclosed
EP-2418190-A1 The method of preparation of enantiomerically enriched products of condensation from racemic acids or acids of the low enentiomeric purity Politechnika Lodzka (PL) 2012-02-15 EP disclosed