SCHEMBL5777920

SCHEMBL5777920

CCNC1Cc2ccc(CCN3CCN(c4snc5ccccc45)CC3)cc2C1(C)C

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 15/20 0.40
HTR2A P28223 14/20 0.40
KCNH2 Q12809 13/20 0.40
DRD2 P14416 11/20 0.40
HTR7 P34969 1/20 0.38
DRD1 P21728 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6402177 0.84 HTR1A (0.57) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL5777922 0.83 HTR1A (0.41) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL6397693 0.80 HTR1A (0.56) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL5738181 0.80 HTR1A (0.44) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL6401301 0.79 HTR1A (0.56) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL6399872 0.75 HTR1A (0.55) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL6399037 0.72 HTR1A (0.68) HTR1AHTR2AKCNH2DRD2
SCHEMBL6401307 0.67 HTR1A (0.59) HTR1AHTR2AKCNH2DRD2HTR7
SCHEMBL22049741 0.67 HTR3A (0.51)
SCHEMBL6398868 0.67 HTR1A (0.67) HTR1AHTR2AKCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697334-A1 HETEROCYCLIC SUBSTITUTED INDANE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA Warner-Lambert Company LLC (US) 2006-09-06 EP disclosed
WO-2005056540-A1 HETEROCYCLIC SUBSTITUTED INDANE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2005-06-23 WO disclosed