SCHEMBL5778029

SCHEMBL5778029

COC(=O)c1ccc(NC(=O)c2cccc(C=Cc3nc(C(C)C)cs3)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.51
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TP53 P04637 2/20 0.48
PKM P14618 1/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48
PLAU P00749 7/20 0.45
PLAT P00750 2/20 0.44
PLG P00747 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
PTPN1 P18031 3/20 0.43
HTT P42858 2/20 0.41
LMNA P02545 2/20 0.41
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5780106 0.90 ALB (0.57) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL27569880 0.90 ALB (0.57) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL5778188 0.79 ALB (0.52) ALBMEN1KMT2ARAB9AALDH1A1
SCHEMBL5779807 0.79 ALB (0.61) ALBPLAUPLAT
SCHEMBL5778350 0.79 ALB (0.57) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL5778781 0.79 ALB (0.55) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL5780400 0.77 ALB (0.53) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL5779175 0.77 ALB (0.55) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL5774563 0.76 ALB (0.69) ALBMEN1KMT2ANPC1RAB9A
SCHEMBL15652097 0.74 RAB9A (0.67) MEN1KMT2ANPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed