SCHEMBL5779141

SCHEMBL5779141

CC1CCN(CCOc2ccc(C(N)=O)cc2)CC1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.63
KDM4E B2RXH2 3/20 0.62
HRH3 Q9Y5N1 10/20 0.61
ALDH1A1 P00352 1/20 0.60
KMT2A Q03164 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3859178 0.99 SIGMAR1 (0.65) SIGMAR1KDM4EHRH3ALDH1A1KMT2A
SCHEMBL22066893 0.88 HRH2 (0.65) SIGMAR1KDM4EHRH3ALDH1A1KMT2A
SCHEMBL30969213 0.85 DRD3 (0.59) KDM4EHRH3ALDH1A1
SCHEMBL3026592 0.84 PSMB1 (0.75) KDM4EHRH3
SCHEMBL30969292 0.83 HRH3 (0.54) HRH3
SCHEMBL30969262 0.83 HRH3 (0.65) KDM4EHRH3
SCHEMBL30969263 0.83 PSMB1 (0.78) KDM4EHRH3ALDH1A1
SCHEMBL3866360 0.81 SIGMAR1 (0.71) SIGMAR1KDM4EHRH3KMT2A
SCHEMBL4022248 0.81 HTR2C (0.54) KDM4EALDH1A1KMT2A
SCHEMBL491570 0.81 HRH3 (0.72) SIGMAR1KDM4EHRH3ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708698-A1 3-(4-PIPERIDINE-1YLMETHYL-PHENYL)-PROPION ACID-PHENYLAMIDE-DERIVATIVES AND RELATED COMPOUNDS USED IN THE FORM OF MCH ANTAGONISTS (MELANINE CONCENTRATING HORMONE) FOR TREATING EATING DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-10-11 EP disclosed
WO-2005063239-A9 3-(4-PIPERIDINE-1YLMETHYL-PHENYL)-PROPION ACID-PHENYLAMIDE-DERIVATIVES AND RELATED COMPOUNDS USED IN THE FORM OF MCH ANTAGONISTS (MELANINE CONCENTRATING HORMONE) FOR TREATING EATING DISORDERS BOEHRINGER INGELHEIM INT (DE) 2006-03-09 WO disclosed
WO-2005063239-A1 3-(4-PIPERIDINE-1YLMETHYL-PHENYL)-PROPION ACID-PHENYLAMIDE-DERIVATIVES AND RELATED COMPOUNDS USED IN THE FORM OF MCH ANTAGONISTS (MELANINE CONCENTRATING HORMONE) FOR TREATING EATING DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-07-14 WO disclosed