SCHEMBL5780643

SCHEMBL5780643

Fc1ccc(-c2c[c]c3ccccc3n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.47
TOP1 P11387 3/20 0.43
ADORA2A P29274 1/20 0.41
MAPK10 P53779 1/20 0.41
MAPK14 Q16539 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TNKS O95271 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
ACP1 P24666 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133411 0.86 DHODH (0.46) TOP1NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL234452 0.85 ACHE (0.47) TOP1RAB9AKDM4ESMN1; SMN2KMT2A
SCHEMBL4901955 0.83 CYP1A1 (0.41) ADORA2ANPC1RAB9AKDM4ETNKS
SCHEMBL4912670 0.83 ALDH1A1 (0.45) ADORA2ANPC1RAB9AKDM4ETNKS
SCHEMBL4907021 0.83 NPC1 (0.53) ADORA2ANPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL5757636 0.82 ADORA2A (0.46) ADORA2AKDM4ESMN1; SMN2ACP1KMT2A
SCHEMBL4875167 0.81 MAPT (0.46) NPC1RAB9AKDM4ESMN1; SMN2KMT2A
SCHEMBL8087264 0.81 CYP2C9 (0.53) MAPK10MAPK14NPC1RAB9AKDM4E
SCHEMBL17941210 0.79 MPO (0.37) NPC1RAB9AKDM4ESMN1; SMN2KMT2A
SCHEMBL4909955 0.79 KDM4E (0.58) ADORA2ANPC1RAB9AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108329297-A Fluorobenzene quinoline substitution carbinol derivatives with anti-tumor activity and its synthetic method and application 河南师范大学 2018-07-27 CN disclosed
EP-1664023-A1 SUSTITUTED ISOQUINOLINE DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2006-06-07 EP disclosed
WO-2005021533-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND METHODS OF USE AMGEN INC (US) 2005-03-10 WO disclosed