SCHEMBL8087264

SCHEMBL8087264

[c]1cc(-c2ccncc2)nc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.53
CYP3A4 P08684 3/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
AR P10275 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
DHODH Q02127 1/20 0.44
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 5/20 0.40
MAPT P10636 4/20 0.40
HPGD P15428 2/20 0.40
NOTUM Q6P988 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.39
RECQL P46063 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL234452 0.87 ACHE (0.47) RAB9ADHODHKDM4EALDH1A1MAPT
SCHEMBL29133411 0.84 DHODH (0.46) NPC1RAB9AARDHODHKDM4E
SCHEMBL4875167 0.82 MAPT (0.46) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL8087285 0.81 CYP19A1 (0.47) CYP2C9CYP3A4NPC1RAB9ACYP1A2
SCHEMBL4907021 0.81 NPC1 (0.53) NPC1RAB9ACYP1A2KDM4EMAPT
SCHEMBL5780643 0.81 CYP19A1 (0.47) NPC1RAB9ADHODHKDM4EALDH1A1
SCHEMBL4912670 0.81 ALDH1A1 (0.45) CYP3A4NPC1RAB9ACYP1A2KDM4E
SCHEMBL4901955 0.81 CYP1A1 (0.41) NPC1RAB9ACYP1A2KDM4EALDH1A1
SCHEMBL8096265 0.79 PDGFRB (0.44) CYP2C9CYP3A4NPC1ARCYP2C19
SCHEMBL4909955 0.77 KDM4E (0.58) NPC1RAB9AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6063956-A APPLYING FUNGICIDE OR INSECTICIDE TO THE LOCUS WHERE CONTROL IS DESIRED ROHM AND HAAS COMPANY (US) 2000-05-16 US disclosed