SCHEMBL578259

SCHEMBL578259

Cc1n[nH]cc1-c1cc(O)nc(-c2nc(C(F)(F)F)cs2)n1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.35
PTGES O14684 2/20 0.34
GFER P55789 1/20 0.32
CYP19A1 P11511 2/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578318 0.86 IDH1 (0.36) IDH1PTGESLMNAPOLB
SCHEMBL578140 0.81 LMNA (0.35) IDH1PTGESLMNAPOLB
SCHEMBL578086 0.80 IDH1 (0.36) IDH1PTGESGFERCYP19A1LMNA
SCHEMBL577784 0.80 IDH1 (0.36) IDH1PTGESGFERCYP19A1LMNA
SCHEMBL11905052 0.79 IDH1 (0.42) IDH1PTGESCYP19A1LMNAPOLB
SCHEMBL577653 0.79 KDM4E (0.37) IDH1PTGESGFERCYP19A1LMNA
SCHEMBL578009 0.79 OPRM1 (0.40) IDH1GFERLMNA
SCHEMBL15215579 0.78 ALDH1A1 (0.43) IDH1PTGESGFERLMNAPOLB
SCHEMBL577698 0.78 PDE10A (0.39) IDH1PTGESLMNAPOLBNTRK1
SCHEMBL577994 0.78 PTGES (0.35) IDH1PTGESCYP19A1LMNANTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2461811-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS USEFUL AGAINST VIRAL INFECTIONS, PARTICULARLY HCV IDENIX Pharmaceuticals, Inc. (US) 2012-06-13 EP disclosed
EP-2417134-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX Pharmaceuticals, Inc. (US) 2012-02-15 EP disclosed
WO-2011017389-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS USEFUL AGAINST VIRAL INFECTIONS, PARTICULARLY HCV IDENIX PHARMACEUTICALS, INC. (US) 2011-02-10 WO disclosed
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed