SCHEMBL5784644

SCHEMBL5784644

Oc1nc(O)c2c(-c3ccccc3)n[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
MAPT P10636 1/20 0.42
GFER P55789 1/20 0.42
KDM4E B2RXH2 3/20 0.41
HPGD P15428 3/20 0.41
MAPK10 P53779 3/20 0.41
GAA P10253 2/20 0.41
TTK P33981 2/20 0.41
ALPL P05186 1/20 0.41
IDO1 P14902 1/20 0.41
RAB9A P51151 3/20 0.39
NPC1 O15118 2/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ALOX15 P16050 1/20 0.38
GRM5 P41594 1/20 0.38
MAP2K4 P45985 2/20 0.36
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5784325 0.84 RAB9A (0.41) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL4930122 0.77 YTHDC1 (0.43) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL5364636 0.73 YTHDC1 (0.43) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL20389460 0.73 MAPK1 (0.42) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL5786736 0.70 ALDH1A1 (0.46) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL15017190 0.70 ADORA3 (0.43) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL12692147 0.69 GRM5 (0.55) GRM5MEN1KMT2AADORA1
SCHEMBL18040266 0.69 DPP4 (0.49) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL15698438 0.69 ALDH1A1 (0.40) ALDH1A1MAPTGFERKDM4EHPGD
SCHEMBL5787312 0.69 HPGD (0.41) ALDH1A1MAPTGFERKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507780-A4 PYRAZOLO-PYRIMIDINE ANILINE COMPOUNDS USEFUL AS KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2006-08-02 EP disclosed
EP-1507780-A1 PYRAZOLO-PYRIMIDINE ANILINE COMPOUNDS USEFUL AS KINASE INHIBITORS Bristol-Myers Squibb Company (US) 2005-02-23 EP disclosed
WO-2003099820-A1 PYRAZOLO-PYRIMIDINE ANILINE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed