SCHEMBL5789324

SCHEMBL5789324

FC(F)(F)c1n[c]c2c(-c3ccccc3)csc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.35
DAPK3 O43293 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
ABL1 P00519 1/20 0.35
NTRK1 P04629 1/20 0.35
LCK P06239 1/20 0.35
CSF1R P07333 1/20 0.35
RET P07949 1/20 0.35
MET P08581 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
PRKACA P17612 1/20 0.35
FLT1 P17948 1/20 0.35
LTK P29376 1/20 0.35
KDR P35968 1/20 0.35
MAP2K2 P36507 1/20 0.35
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
CSNK1A1 P48729 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6364382 0.78 ESR1 (0.45) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL6362941 0.74 MAPT (0.38) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL6359795 0.74 ALDH1A1 (0.42) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL2368948 0.74 ALDH1A1 (0.38) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL2368688 0.74 FGFR1 (0.40) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL6359338 0.72 ESR1 (0.38) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL2369443 0.71 ALDH1A1 (0.55) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL6359949 0.70 SQOR (0.37) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL5790639 0.69 HTT (0.35) FGFR1DAPK3PRKD3MAP4K4ABL1
SCHEMBL5791688 0.69 LMNA (0.52) ALDH1A1RAB9ALMNANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641803-A1 THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS Xention Discovery Limited (GB) 2006-04-05 EP disclosed
WO-2004111057-A1 THIENOPYRIMIDINE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS XENTION DISCOVERY LIMITED (GB) 2004-12-23 WO disclosed