SCHEMBL5791587

SCHEMBL5791587

CC(C)CNN(C(=O)CCC1CCCC1)c1ccnc(C#N)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
TP53 P04637 2/20 0.36
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CTSK P43235 5/20 0.36
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
ATM Q13315 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CTSS P25774 3/20 0.34
CTSL P07711 1/20 0.34
OPRM1 P35372 2/20 0.34
OPRL1 P41146 2/20 0.34
FGFR4 P22455 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5807653 0.82 CTSK (0.35) CTSKFGFR4
SCHEMBL5793909 0.79 CTSK (0.41) CTSKFGFR4GPR119
SCHEMBL5791458 0.78 KMT2A (0.41) MEN1KMT2ANPC1RAB9ATP53
SCHEMBL5794212 0.77 HPGD (0.41) MEN1KMT2ARAB9ASMN1; SMN2CTSK
SCHEMBL5793159 0.75 CTSK (0.36) KMT2ANPC1RAB9ASMN1; SMN2CTSK
SCHEMBL5791288 0.75 MAPK14 (0.43) NPC1RAB9ATSHRCTSKFGFR4
Trifluoroacetic Acid SCHEMBL5793434 0.75 CTSK (0.44) MEN1KMT2ACTSKCTSSCTSL
SCHEMBL5791044 0.74 CTSK (0.45) CTSKCTSSCTSLFGFR4
Trifluoroacetic Acid SCHEMBL5791892 0.72 CTSK (0.38) CTSKCTSSFGFR4
SCHEMBL5792335 0.72 CTSK (0.37) KMT2ANPC1RAB9ATSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed