SCHEMBL5793159

SCHEMBL5793159

CC(C)CNN(C(=O)Cc1ccc(N(C)C)cc1)c1ccnc(C#N)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.36
FGFR4 P22455 1/20 0.35
CACNA1G O43497 3/20 0.35
CACNA1H O95180 3/20 0.35
CACNA1I Q9P0X4 3/20 0.35
KMT2A Q03164 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PANK3 Q9H999 1/20 0.33
ACACB O00763 1/20 0.32
GPR4 P46093 1/20 0.32
HDAC1 Q13547 1/20 0.32
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
MCL1 Q07820 1/20 0.31
CNR2 P34972 1/20 0.31
CTSL P07711 1/20 0.31
CTSB P07858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5794212 0.90 HPGD (0.41) CTSKFGFR4KMT2ARAB9ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5793434 0.83 CTSK (0.44) CTSKFGFR4KMT2ACTSLCTSS
SCHEMBL5792562 0.79 CTSK (0.45) CTSKFGFR4KMT2ARAB9AALDH1A1
SCHEMBL8270011 0.79 ALDH1A1 (0.39) CTSKFGFR4CACNA1GCACNA1HCACNA1I
SCHEMBL5807653 0.78 CTSK (0.35) CTSKFGFR4GPR4
SCHEMBL5793909 0.78 CTSK (0.41) CTSKFGFR4GPR4
Trifluoroacetic Acid SCHEMBL5791291 0.77 CTSK (0.38) CTSKKMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL5808749 0.76 CACNA1G (0.37) CTSKFGFR4CACNA1GCACNA1HCACNA1I
SCHEMBL5791288 0.76 MAPK14 (0.43) CTSKFGFR4NPC1RAB9A
SCHEMBL5791587 0.75 MEN1 (0.36) CTSKFGFR4KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed