SCHEMBL5791973

SCHEMBL5791973

CC(C)(C)c1ccc(CN2CCC(C(=O)O)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
S1PR5 Q9H228 6/20 0.57
S1PR4 O95977 4/20 0.57
S1PR1 P21453 4/20 0.57
S1PR3 Q99500 2/20 0.53
HRH3 Q9Y5N1 1/20 0.52
CACNA1G O43497 2/20 0.51
LTA4H P09960 2/20 0.50
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR2B P41595 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
MAPT P10636 1/20 0.49
RAB9A P51151 1/20 0.49
TEAD1 P28347 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15942972 0.92 S1PR5 (0.63) MEN1KMT2AS1PR5S1PR4S1PR1
SCHEMBL798026 0.88 MEN1 (0.56) MEN1KMT2AS1PR5S1PR4S1PR1
SCHEMBL15942971 0.86 SIGMAR1 (0.57) MEN1KMT2AS1PR5S1PR4S1PR1
SCHEMBL24529849 0.85 SIGMAR1 (0.62) S1PR5HRH3KDM4EALDH1A1SIGMAR1
SCHEMBL13242411 0.85 S1PR5 (0.74) S1PR5S1PR4S1PR1S1PR3
SCHEMBL7238102 0.84 MEN1 (0.62) MEN1KMT2AS1PR5CACNA1GSIGMAR1
SCHEMBL13236630 0.83 S1PR5 (0.66) S1PR5S1PR4S1PR1S1PR3HRH3
SCHEMBL797736 0.83 S1PR1 (0.54) MEN1KMT2AS1PR5S1PR4S1PR1
SCHEMBL2073212 0.81 DRD2 (0.60) MEN1KMT2AS1PR5HRH3KDM4E
SCHEMBL12412709 0.81 ALDH1A1 (0.59) MEN1KMT2AHRH3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8802663-B2 Pyrazole oxadiazole derivatives as S1P1 agonists MERCK SERONO SA (CH) 2014-08-12 US disclosed
WO-2006002956-A1 PIPERIDINE DERIVATIVES AND THEIR USE AS GLYCINE TRANSPORTER INHIBITORS GLAXO GROUP LIMITED (GB) 2006-01-12 WO disclosed
WO-2006002956-A1 PIPERIDINE DERIVATIVES AND THEIR USE AS GLYCINE TRANSPORTER INHIBITORS GLAXO GROUP LIMITED (GB) 2006-01-12 WO disclosed