SCHEMBL5792191

SCHEMBL5792191

CC(C)CN(NC(=O)Cc1ccc(OC(F)(F)F)cc1)c1ccnc(C#N)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WNT3A P56704 1/20 0.38
CACNA1H O95180 3/20 0.38
CACNA1G O43497 2/20 0.38
CACNA1I Q9P0X4 2/20 0.38
EPHX2 P34913 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NTRK1 P04629 1/20 0.37
NLRP3 Q96P20 1/20 0.36
CTSK P43235 3/20 0.36
ACACB O00763 1/20 0.36
LTA4H P09960 1/20 0.36
PANK3 Q9H999 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
MAPK8 P45983 1/20 0.35
VNN1 O95497 1/20 0.35
CCNA2 P20248 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5794190 0.89 ALDH1A1 (0.41) WNT3AMEN1KMT2ASMN1; SMN2CTSK
SCHEMBL5794599 0.88 CTSK (0.38) CACNA1HNTRK1CTSKCTSLCTSB
SCHEMBL5790864 0.87 HTT (0.39) WNT3AKMT2ACTSKCTSLCTSB
SCHEMBL5804787 0.86 HPGD (0.41) WNT3ASMN1; SMN2CTSKCTSLCTSB
Trifluoroacetic Acid SCHEMBL5791900 0.85 CTSK (0.44) KMT2ASMN1; SMN2CTSKCTSLCTSB
SCHEMBL8270730 0.85 CTSK (0.42) MEN1KMT2ASMN1; SMN2CTSKCTSL
SCHEMBL8270011 0.85 ALDH1A1 (0.39) CACNA1HCACNA1GCACNA1IKMT2ACTSK
SCHEMBL5794156 0.85 CTSK (0.40) KMT2ASMN1; SMN2CTSKCTSLCTSB
Trifluoroacetic Acid SCHEMBL5790897 0.85 CTSK (0.38) MEN1KMT2ASMN1; SMN2CTSKCTSL
SCHEMBL8271456 0.85 CTSK (0.47) KMT2ASMN1; SMN2CTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed