SCHEMBL5794599

SCHEMBL5794599

CC(C)CN(NC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccnc(C#N)n1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
ANO1 Q5XXA6 1/20 0.38
MAPK8 P45983 1/20 0.37
MAPK10 P53779 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
MMP3 P08254 1/20 0.36
CNR2 P34972 2/20 0.35
UTS2R Q9UKP6 3/20 0.35
P2RX7 Q99572 1/20 0.35
MCHR1 Q99705 2/20 0.35
CACNA1H O95180 1/20 0.35
NTRK1 P04629 1/20 0.34
RIOK2 Q9BVS4 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5790864 0.89 HTT (0.39) CTSKCTSLCTSBCTSSANO1
SCHEMBL8270502 0.89 ANO1 (0.42) CTSKANO1P2RX7RIOK2
SCHEMBL5804787 0.88 HPGD (0.41) CTSKCTSLCTSBCTSSANO1
SCHEMBL5792191 0.88 WNT3A (0.38) CTSKCTSLCTSBCTSSMAPK8
Trifluoroacetic Acid SCHEMBL5791900 0.88 CTSK (0.44) CTSKCTSLCTSBCTSSMAPK8
SCHEMBL8270011 0.87 ALDH1A1 (0.39) CTSKCTSLCTSBCTSSHDAC1
SCHEMBL8270730 0.87 CTSK (0.42) CTSKCTSLCTSBCTSS
SCHEMBL8269396 0.87 CTSK (0.45) CTSKCTSLCTSBCTSSMMP3
SCHEMBL5794156 0.87 CTSK (0.40) CTSKCTSLCTSBCTSSMAPK8
Trifluoroacetic Acid SCHEMBL5790897 0.87 CTSK (0.38) CTSKCTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed