SCHEMBL5793302

SCHEMBL5793302

O=CCc1ccccc1OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.46
SLC1A5 Q15758 1/20 0.45
PTPN1 P18031 4/20 0.43
PTPN2 P17706 3/20 0.43
PTPN6 P29350 3/20 0.43
PTPRC P08575 1/20 0.43
PTPRB P23467 1/20 0.43
PTPN11 Q06124 1/20 0.43
IDO1 P14902 2/20 0.41
CACNA1F O60840 1/20 0.41
CACNA1D Q01668 1/20 0.41
CACNA1S Q13698 1/20 0.41
CACNA1C Q13936 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
HIF1A Q16665 1/20 0.40
PPARG P37231 1/20 0.40
PTGER1 P34995 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HTR1A P08908 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18002778 0.87 PTPN1 (0.54) PTPN1PTPN2PTPN6PTPRCPTPRB
SCHEMBL23673331 0.80 ALDH1A1 (0.53) TACR1PTPN1PTPN2PTPN6PTPRC
SCHEMBL17141460 0.80 HTR2C (0.51) SLC1A5PTPN1PTPN2PTPN6PTPRC
SCHEMBL872421 0.79 HTR1A (0.61) PTGER1POLBMAPTHTR1ADRD2
SCHEMBL12247630 0.78 ABCB1 (0.43) TACR1SLC1A5PTGER1MAPTHTR1A
SCHEMBL16406686 0.77 PTPRC (0.45) SLC1A5PTPN1PTPN2PTPN6PTPRC
SCHEMBL23683173 0.76 LMNA (0.63) TACR1
SCHEMBL8507790 0.75 TACR1 (0.49) TACR1IDO1CACNA1FCACNA1DCACNA1S
SCHEMBL9435408 0.75 SLC1A5 (0.43) TACR1SLC1A5PTPN1PTGER1HTR1A
SCHEMBL18002701 0.74 POLB (0.49) TACR1PTPN1PTPN2PTPN6PTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006014942-A1 ARYLOXYALKYLAMINE NK-1/SSRI INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-09 WO disclosed