SCHEMBL5795537

SCHEMBL5795537

CCCCCCCn1cc(C2=CCN(C(=O)OC(C)(C)C)CC2)c2cc(-c3c(CC)cccc3CC)ncc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.46
HTR6 P50406 1/20 0.45
SCN9A Q15858 1/20 0.44
GRM1 Q13255 10/20 0.43
GRM5 P41594 9/20 0.43
EED O75530 1/20 0.41
RBBP4 Q09028 1/20 0.41
SUZ12 Q15022 1/20 0.41
EZH2 Q15910 1/20 0.41
WNT3A P56704 1/20 0.40
BRD4 O60885 1/20 0.39
DGAT2 Q96PD7 1/20 0.39
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1762832 0.84 PDK4 (0.49) PDK4HTR6SCN9AGRM1GRM5
SCHEMBL5798518 0.81 ALDH1A1 (0.43) SCN9A
SCHEMBL1762815 0.79 GABRP (0.54) PDK4HTR6GRM1GRM5EED
SCHEMBL18409265 0.70 GRM1 (0.52) PDK4GRM1GRM5WNT3A
SCHEMBL14540703 0.69 HTR6 (0.70) PDK4HTR6SCN9AGRM1GRM5
SCHEMBL18409268 0.68 GRM1 (0.52) PDK4GRM1GRM5WNT3A
SCHEMBL8026743 0.67 HTR6 (0.67) PDK4HTR6SCN9AGRM1GRM5
SCHEMBL20030944 0.67 SCN9A (0.49) PDK4HTR6SCN9AGRM1GRM5
SCHEMBL19092559 0.67 PDK4 (0.58) PDK4HTR6SCN9AGRM1GRM5
SCHEMBL15167555 0.66 GRM1 (0.57) PDK4HTR6GRM1GRM5WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006042102-A2 PYRROLO-PYRIDINE, PYRROLO-PYRIMIDINE AND RELATED HETEROCYCLIC COMPOUNDS NEUROGEN CORPORATION (US) 2006-04-20 WO disclosed