SCHEMBL5795648

SCHEMBL5795648

CC(CCC(N)=O)CNC(C(=O)OC(C)(C)C)c1ccc2[nH]ccc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
MAOA P21397 2/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
NR3C1 P04150 1/20 0.33
ADRB1 P08588 1/20 0.32
HDAC1 Q13547 2/20 0.32
TGFBR1 P36897 1/20 0.32
AURKA O14965 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795781 0.86 PTGS2 (0.38) PTGS2MAOA
SCHEMBL5795645 0.77 TAS1R3 (0.48) PTGS2TAS1R3TAS1R1MAOASLC6A2
SCHEMBL5795647 0.77 TAS1R3 (0.48) PTGS2TAS1R3TAS1R1MAOASLC6A2
SCHEMBL7214901 0.73 PTGS2 (0.45) PTGS2TAS1R3TAS1R1MAOASLC6A2
SCHEMBL10631836 0.69 PTGS2 (0.47) PTGS2TAS1R3TAS1R1MAOASLC6A2
SCHEMBL2307317 0.66 SLC6A2 (0.53) PTGS2SLC6A2SLC6A4SLC6A3NR3C1
SCHEMBL30795530 0.65 PTGS2 (0.49) PTGS2MAOASLC6A2SLC6A4SLC6A3
SCHEMBL15324491 0.64 MAOA (0.42) PTGS2TAS1R3TAS1R1MAOASLC6A2
SCHEMBL3106353 0.64 TUBB4A (0.51) TAS1R3TAS1R1MAOACTNNB1WNT3A
Hydrochloric Acid SCHEMBL16583860 0.64 MAOA (0.42) PTGS2TAS1R3TAS1R1MAOASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006034480-A2 SULFONAMIDE BICYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-03-30 WO disclosed