SCHEMBL5797285

SCHEMBL5797285

COc1cc2c(C(C(=O)O)C(C)(C)C)c(C)n(C(=S)c3ccc(C)cc3)c2cc1F.COc1cc2c(CC(=O)O)c(C)n(C(=S)c3ccc(C)cc3)c2cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.45
PTGS2 P35354 2/20 0.45
AKR1C3 P42330 11/20 0.44
AKR1C2 P52895 10/20 0.44
ABCB1 P08183 3/20 0.38
LMNA P02545 3/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 3/20 0.38
NPSR1 Q6W5P4 3/20 0.38
CYP2D6 P10635 2/20 0.38
HIF1A Q16665 2/20 0.38
AKR1C4 P17516 2/20 0.38
AKR1C1 Q04828 2/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.38
KDM4E B2RXH2 2/20 0.38
PMP22 Q01453 2/20 0.38
MEN1 O00255 1/20 0.38
PTGES O14684 1/20 0.38
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6425829 0.92 RAB9A (0.34) PTGS1PTGS2AKR1C3AKR1C2LMNA
SCHEMBL5558645 0.89 AKR1C3 (0.54) PTGS1PTGS2AKR1C3AKR1C2ABCB1
SCHEMBL5800524 0.87 AKR1C3 (0.50) PTGS1PTGS2AKR1C3AKR1C2ABCB1
SCHEMBL5799879 0.85 PTGS2 (0.43) PTGS1PTGS2AKR1C3AKR1C2ABCB1
SCHEMBL6423578 0.83 PTGS1 (0.41) PTGS1PTGS2AKR1C3AKR1C2ABCB1
SCHEMBL5798139 0.82 PTGS1 (0.42) PTGS1PTGS2AKR1C3AKR1C2ABCB1
SCHEMBL5797328 0.82 PTGS1 (0.69) PTGS1PTGS2AKR1C3AKR1C2ABCB1
SCHEMBL6424686 0.82 PTGS1 (0.44) PTGS1PTGS2AKR1C3AKR1C2RAB9A
SCHEMBL6424402 0.81 LMNA (0.37) PTGS1PTGS2AKR1C3AKR1C2LMNA
SCHEMBL6425557 0.81 LMNA (0.35) PTGS1PTGS2AKR1C3AKR1C2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed