SCHEMBL5797476

SCHEMBL5797476

Cc1c(-c2ccccc2)[c]ccc1-c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2E1 P05181 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PARP11 Q9NR21 1/20 0.42
CYP11B1 P15538 4/20 0.41
CYP11B2 P19099 4/20 0.41
GPR35 Q9HC97 2/20 0.41
PTGS2 P35354 1/20 0.40
NPY5R Q15761 1/20 0.40
ALK Q9UM73 1/20 0.40
CYP19A1 P11511 2/20 0.39
CYP17A1 P05093 1/20 0.39
KCNA5 P22460 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28592408 0.79 CYP2A6 (0.47) CYP2A6CYP3A4CYP2E1CYP2D6CYP2C9
SCHEMBL21742825 0.76 PTGS2 (0.54) CYP2A6CYP3A4CYP2E1CYP2D6CYP2C9
SCHEMBL5796609 0.75 KDM4E (0.39) CYP2A6ALDH1A1CYP1A2NPY5R
SCHEMBL21742648 0.72 PARP10 (0.48) CYP2A6CYP3A4CYP2E1CYP2D6CYP2C9
SCHEMBL9958033 0.72 ALDH1A1 (0.47) CYP2A6CYP3A4CYP2C9CYP2B6CYP2C19
SCHEMBL10416386 0.72 MAPT (0.40) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL23071560 0.71 CYP2A6 (0.50) CYP2A6CYP3A4CYP2E1CYP2D6CYP2C9
SCHEMBL21742767 0.70 CYP2A6 (0.54) CYP2A6CYP3A4CYP2E1CYP2D6CYP2C9
SCHEMBL8879482 0.70 CYP2A6 (0.49) CYP2A6CYP3A4CYP2E1CYP2D6CYP2C9
SCHEMBL982200 0.70 ALDH1A1 (0.33) CYP2A6CYP2B6ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006033995-A2 THIAZOLIDIN-4-ONES HAVING ANTI-HEPATITIS B ACTIVITY VALEANT RESEARCH AND DEVELOPMENT (US) 2006-03-30 WO disclosed