SCHEMBL5797987

SCHEMBL5797987

NC(=O)c1nc2cccnc2s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.54
LIMK1 P53667 2/20 0.47
IKBKB O14920 1/20 0.47
CHUK O15111 1/20 0.47
CYP2C9 P11712 1/20 0.44
POLB P06746 2/20 0.44
NPC1 O15118 8/20 0.43
RAB9A P51151 7/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
PARP1 P09874 1/20 0.41
MAPT P10636 5/20 0.40
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 4/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TP53 P04637 2/20 0.40
ATM Q13315 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30943923 0.84 PDK1 (0.56) PDK1CYP2C9POLBNPC1RAB9A
SCHEMBL2645378 0.84 PDK1 (0.56) PDK1CYP2C9POLBNPC1RAB9A
SCHEMBL24960020 0.79 ALDH1A1 (0.60) PDK1CYP2C9POLBNPC1RAB9A
SCHEMBL9212502 0.75 PDK1 (0.58) PDK1POLBNPC1RAB9ASMN1; SMN2
SCHEMBL16264455 0.75 CYP2C9 (0.58) PDK1CYP2C9POLBNPC1RAB9A
SCHEMBL2902912 0.74 MAPT (0.54) POLBNPC1RAB9ASMN1; SMN2PARP1
Hydrochloric Acid SCHEMBL2905808 0.73 MAPT (0.53) POLBNPC1RAB9ASMN1; SMN2PARP1
SCHEMBL369480 0.73 ALDH1A1 (0.62) PDK1POLBNPC1RAB9ASMN1; SMN2
SCHEMBL20505867 0.72 DYRK1A (0.34) LIMK1IKBKBTSHR
SCHEMBL15109690 0.72 LIMK1 (0.47) LIMK1IKBKBCHUKPARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074089-B1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2013-09-18 EP claimed
WO-2006071035-A1 NOVEL ([1,3]THIAZOLO[5,4-B]PYRIDIN-2-YL)-2-CARBOXAMIDE DERIVATIVES LG LIFE SCIENCES, LTD. (KR) 2006-07-06 WO disclosed