SCHEMBL5800380

SCHEMBL5800380

N#CC1(NC(=O)C(Cc2cc(I)c(O)c(I)c2)NC(=O)c2ccc(N3CCN(C4CC4)CC3)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSL P07711 17/20 0.52
CTSS P25774 11/20 0.52
CTSB P07858 9/20 0.52
CTSK P43235 9/20 0.52
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6403855 0.88 CTSL (0.55) CTSLCTSSCTSBCTSKCYP2D6
SCHEMBL6403849 0.88 CTSL (0.55) CTSLCTSSCTSBCTSKCYP2D6
SCHEMBL5801033 0.87 CTSK (0.49) CTSLCTSSCTSBCTSK
SCHEMBL5797321 0.84 POLB (0.45)
SCHEMBL5808560 0.83 ADRB3 (0.46)
SCHEMBL5800383 0.82 CTSK (0.45) CTSLCTSSCTSBCTSK
Lithium Ion SCHEMBL5808563 0.82 MEN1 (0.41) CTSK
SCHEMBL5812496 0.81 CTSK (0.47) CTSLCTSSCTSBCTSK
SCHEMBL6208313 0.74 CTSL (0.53) CTSLCTSSCTSBCTSK
SCHEMBL6208306 0.74 CTSL (0.53) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006042103-A2 REVERSIBLE INHIBITORS OF CATHEPSIN B AXYS PHARMACEUTICALS, INC. (US) 2006-04-20 WO claimed
WO-2006042103-A2 REVERSIBLE INHIBITORS OF CATHEPSIN B AXYS PHARMACEUTICALS, INC. (US) 2006-04-20 WO disclosed