SCHEMBL5800501

SCHEMBL5800501

CC(=O)CN(c1cc[c]cc1)c1ccc(C)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 5/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TSHR P16473 1/20 0.33
HPGD P15428 1/20 0.33
LMNA P02545 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HTT P42858 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6417145 0.76 ALDH1A1 (0.39) ALDH1A1TSHRLMNAHTTTDP1
SCHEMBL11560187 0.74 ALDH1A1 (0.46) KEAP1NFE2L2RAB9AALDH1A1SMN1; SMN2
SCHEMBL12419483 0.72 ESR1 (0.44) TSHRTDP1CES2CES1
SCHEMBL374605 0.71 MTNR1A (0.53) RAB9AALDH1A1SMN1; SMN2TSHRLMNA
SCHEMBL125310 0.71 ALDH1A1 (0.46) ALDH1A1TSHRKDM4ETDP1
SCHEMBL11318899 0.71 KEAP1 (0.41) KEAP1NFE2L2RAB9AALDH1A1SMN1; SMN2
SCHEMBL3105534 0.70 MTNR1A (0.52) RAB9AALDH1A1SMN1; SMN2TSHRLMNA
SCHEMBL16573331 0.69 KEAP1 (0.40) KEAP1NFE2L2RAB9AALDH1A1SMN1; SMN2
SCHEMBL9632432 0.69 KEAP1 (0.51) KEAP1NFE2L2RAB9ASMN1; SMN2TSHR
SCHEMBL9461590 0.68 ALDH1A1 (0.48) KEAP1NFE2L2RAB9AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641762-A2 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2006-04-05 EP disclosed
WO-2005005393-A2 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-01-20 WO disclosed