SCHEMBL5801129

SCHEMBL5801129

CC(NC(=O)N1CCC2(CC1)C(=O)N(C)CN2c1ccccc1)C(NC(=O)c1c(Cl)cccc1Cl)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 7/20 0.55
OPRM1 P35372 11/20 0.46
OPRK1 P41145 11/20 0.46
OPRL1 P41146 11/20 0.46
OPRD1 P41143 9/20 0.46
CCR3 P51677 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2A P28223 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801972 0.89 OPRM1 (0.51) OPRM1OPRK1OPRL1OPRD1
SCHEMBL5803270 0.88 OPRM1 (0.46) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL5802736 0.86 OPRM1 (0.49) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL5783277 0.84 ENPP2 (0.49) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL6632197 0.83 ENPP2 (0.49) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL5950765 0.82 ENPP2 (0.50) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL6629784 0.81 ENPP2 (0.51) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL6481441 0.81 ENPP2 (0.47) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL5802411 0.80 ENPP2 (0.46) ENPP2OPRM1OPRK1OPRL1OPRD1
SCHEMBL5799004 0.79 ENPP2 (0.50) ENPP2OPRM1OPRK1OPRL1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329451-B1 SPIRO COMPOUNDS AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES (JP) 2006-08-23 EP disclosed
EP-1329451-A1 SPIRO COMPOUNDS AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-23 EP disclosed