SCHEMBL5801186

SCHEMBL5801186

CC(C)(C)c1ccc(C2CC2CO)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 13/20 0.49
HTR2B P41595 11/20 0.44
HTR2A P28223 7/20 0.44
CNR2 P34972 4/20 0.43
KDM1A O60341 1/20 0.42
SLC6A2 P23975 3/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
MAOB P27338 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9820788 0.81 HTR2C (0.49) HTR2CHTR2BHTR2AKDM1ASLC6A2
SCHEMBL11965119 0.79 HTR2C (0.63) HTR2CHTR2BHTR2ASLC6A2SLC6A4
SCHEMBL11902887 0.79 HTR2C (0.63) HTR2CHTR2BHTR2ASLC6A2SLC6A4
SCHEMBL22436649 0.76 SLC6A2 (0.45) HTR2CCNR2KDM1ASLC6A2SLC6A4
SCHEMBL9820835 0.76 HTR2C (0.41) HTR2CHTR2BHTR2AKDM1AMAOB
SCHEMBL16585035 0.75 HTR2C (0.66) HTR2CHTR2BHTR2AKDM1ASLC6A2
SCHEMBL17080568 0.75 HTR2C (0.41) HTR2CHTR2BHTR2ASLC6A2SLC6A4
SCHEMBL4893904 0.75 HTR2C (0.66) HTR2CHTR2BHTR2AKDM1ASLC6A2
SCHEMBL16569276 0.75 HTR2C (0.41) HTR2CHTR2BHTR2ASLC6A2SLC6A4
SCHEMBL13591154 0.75 HTR2C (0.63) HTR2CHTR2BHTR2ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006098554-A1 NOVEL COMPOUNDS, ISOMER THEREOF OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST; AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2006-09-21 WO disclosed
EP-0188887-B1 TERTIARY AMINE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-05-02 EP disclosed
EP-0188887-A1 Tertiary amine compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-07-30 EP disclosed