SCHEMBL5801541

SCHEMBL5801541

CCC(OC)c1cccc(C#N)c1N

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
AOC3 Q16853 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 2/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.32
GAA P10253 2/20 0.31
POLB P06746 1/20 0.31
MAP2K1 Q02750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19779659 0.80 TSHR (0.39) ALDH1A1L3MBTL1KDM4ETSHRMAP2K1
SCHEMBL20621249 0.79 TSHR (0.43) ALDH1A1L3MBTL1KDM4EUSP2TSHR
SCHEMBL26596713 0.79 ALDH1A1 (0.35) ALDH1A1L3MBTL1KDM4EUSP2TSHR
SCHEMBL5801533 0.78 CYP1A2 (0.36) ALDH1A1KDM4EUSP2TSHRGAA
SCHEMBL7645209 0.76 ALDH1A1 (0.37) ALDH1A1L3MBTL1KDM4EUSP2TSHR
SCHEMBL19768970 0.74 GABRA1 (0.40) ALDH1A1L3MBTL1TSHRPOLBMAP2K1
SCHEMBL84270 0.71 TSHR (0.36) ALDH1A1L3MBTL1TSHRMAP2K1
SCHEMBL4542360 0.69 IKBKB (0.34) KDM4E
SCHEMBL19734472 0.69 MAOB (0.34) TSHR
SCHEMBL2423501 0.69 TSHR (0.46) ALDH1A1KDM4EUSP2TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385524-A4 PYRAZOLOPYRIMIDINES AS THERAPEUTIC AGENTS ABBOTT GMBH & CO KG (DE) 2006-02-01 EP disclosed
EP-1385524-A1 PYRAZOLOPYRIMIDINES AS THERAPEUTIC AGENTS Abbott GmbH & Co. KG (DE) 2004-02-04 EP disclosed
WO-2002080926-A1 PYRAZOLOPYRIMIDINES AS THERAPEUTIC AGENTS ABBOTT GMBH & CO. KG (DE) 2002-10-17 WO disclosed