SCHEMBL5804885

SCHEMBL5804885

Cc1cc(N(CC(C)C)NC(=O)OC(C)(C)C)nc(Cl)n1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
AAK1 Q2M2I8 13/20 0.36
THRB P10828 1/20 0.33
STK17B O94768 1/20 0.33
STK17A Q9UEE5 1/20 0.33
PTGER1 P34995 1/20 0.33
NPR3 P17342 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306751 0.91 STK17B (0.37) AAK1STK17BSTK17ANPR3CA12
SCHEMBL5305779 0.86 AAK1 (0.36) AAK1STK17BSTK17ANPR3CA12
SCHEMBL5794142 0.86 MEN1 (0.40) MEN1KMT2AAAK1THRBSTK17B
SCHEMBL5306992 0.85 ATR (0.36) AAK1STK17BSTK17ANPR3CA12
SCHEMBL5791173 0.83 GPR119 (0.39) AAK1
SCHEMBL8140939 0.81 AAK1 (0.47) AAK1STK17BSTK17A
SCHEMBL5792631 0.76 STK17B (0.42) AAK1STK17BSTK17A
SCHEMBL5306935 0.76 AAK1 (0.36) AAK1STK17BSTK17ANPR3
SCHEMBL5306326 0.74 STK17B (0.47) AAK1STK17BSTK17A
SCHEMBL5370705 0.73 MAPT (0.41) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed