SCHEMBL5306992

SCHEMBL5306992

COC(=O)c1cc(N(CC(C)C)NC(=O)OC(C)(C)C)nc(Cl)n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.36
AAK1 Q2M2I8 10/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
ABCB1 P08183 3/20 0.32
TRPA1 O75762 1/20 0.32
STK17B O94768 1/20 0.32
STK17A Q9UEE5 1/20 0.32
NPR3 P17342 1/20 0.32
NQO2 P16083 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306751 0.88 STK17B (0.37) AAK1CA12CA1CA2CA9
SCHEMBL5305779 0.86 AAK1 (0.36) ATRAAK1CA12CA1CA2
SCHEMBL5804885 0.85 MEN1 (0.38) AAK1CA12CA1CA2CA9
SCHEMBL5311129 0.84 LMNA (0.34) ATRAAK1ABCB1TRPA1
SCHEMBL8140939 0.79 AAK1 (0.47) ATRAAK1TRPA1STK17BSTK17A
SCHEMBL5454475 0.73 AAK1 (0.34) AAK1TRPA1
SCHEMBL5306326 0.72 STK17B (0.47) ATRAAK1TRPA1STK17BSTK17A
SCHEMBL5309237 0.72 STK17B (0.40) ATRAAK1TRPA1STK17BSTK17A
SCHEMBL5791173 0.72 GPR119 (0.39) AAK1TRPA1
SCHEMBL5794142 0.71 MEN1 (0.40) ATRAAK1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed