SCHEMBL5305779

SCHEMBL5305779

COc1cc(N(CC(C)C)NC(=O)OC(C)(C)C)nc(Cl)n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 10/20 0.36
AR P10275 1/20 0.35
SUV39H2 Q9H5I1 1/20 0.33
STK17B O94768 1/20 0.32
STK17A Q9UEE5 1/20 0.32
ATR Q13535 1/20 0.32
ABCB1 P08183 1/20 0.32
NPR3 P17342 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306751 0.89 STK17B (0.37) AAK1STK17BSTK17ANPR3CA12
SCHEMBL5804885 0.86 MEN1 (0.38) AAK1STK17BSTK17ANPR3CA12
SCHEMBL5306992 0.86 ATR (0.36) AAK1STK17BSTK17AATRABCB1
SCHEMBL5454475 0.85 AAK1 (0.34) AAK1AR
SCHEMBL8140939 0.80 AAK1 (0.47) AAK1STK17BSTK17AATR
SCHEMBL5309237 0.75 STK17B (0.40) AAK1STK17BSTK17AATR
SCHEMBL5794142 0.74 MEN1 (0.40) AAK1STK17BSTK17AATRCA12
SCHEMBL5306326 0.73 STK17B (0.47) AAK1STK17BSTK17AATR
SCHEMBL5791173 0.72 GPR119 (0.39) AAK1
SCHEMBL5311129 0.72 LMNA (0.34) AAK1ATRABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed