SCHEMBL5306751

SCHEMBL5306751

CC(C)CN(NC(=O)OC(C)(C)C)c1cc(Cl)nc(Cl)n1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
STK17B O94768 1/20 0.37
STK17A Q9UEE5 1/20 0.37
AAK1 Q2M2I8 13/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
NPR3 P17342 1/20 0.34
AKT1 P31749 2/20 0.33
TRPA1 O75762 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5804885 0.91 MEN1 (0.38) STK17BSTK17AAAK1CA12CA1
SCHEMBL5305779 0.89 AAK1 (0.36) STK17BSTK17AAAK1CA12CA1
SCHEMBL5306992 0.88 ATR (0.36) STK17BSTK17AAAK1CA12CA1
SCHEMBL8140939 0.83 AAK1 (0.47) STK17BSTK17AAAK1TRPA1
SCHEMBL5306326 0.76 STK17B (0.47) STK17BSTK17AAAK1TRPA1
SCHEMBL5791173 0.76 GPR119 (0.39) AAK1TRPA1
SCHEMBL5794142 0.76 MEN1 (0.40) STK17BSTK17AAAK1CA12CA1
SCHEMBL5306935 0.75 AAK1 (0.36) STK17BSTK17AAAK1NPR3AKT1
SCHEMBL5792631 0.75 STK17B (0.42) STK17BSTK17AAAK1TRPA1
SCHEMBL5454475 0.75 AAK1 (0.34) AAK1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed