SCHEMBL5807345

SCHEMBL5807345

CCOC(=O)Oc1cc2cc(Oc3ccc(Nc4nc5cc(C(F)(F)F)cc(Cl)c5[nH]4)cc3)ccc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 6/20 0.42
BRAF P15056 4/20 0.42
KDR P35968 10/20 0.40
TEK Q02763 8/20 0.40
BRD4 O60885 1/20 0.36
LGALS8 O00214 1/20 0.35
LGALS3 P17931 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5453152 0.88 KDM4E (0.46) RAF1BRAFKDRTEKLGALS8
SCHEMBL5444098 0.79 KDM4E (0.46) RAF1BRAFKDRTEKLGALS8
SCHEMBL14627466 0.77 RAF1 (0.38) RAF1BRAFKDRTEK
SCHEMBL5796359 0.76 PTGES (0.40) RAF1BRAFKDRTEK
SCHEMBL5450095 0.72 KDR (0.44) RAF1BRAFKDRTEK
SCHEMBL5796233 0.71 BRAF (0.36) RAF1BRAFKDRTEK
SCHEMBL14521447 0.71 POLB (0.41) KDRALDH1A1
SCHEMBL5456884 0.71 NPC1 (0.46) RAF1BRAFKDRTEKALDH1A1
SCHEMBL5447398 0.70 PTGES (0.40) RAF1BRAFKDRTEK
SCHEMBL5795361 0.70 RIPK1 (0.41) RAF1BRAFKDRTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656377-A1 AMINOBENZIMIDAZOLE DERIVATIVES MERCK PATENT GmbH (DE) 2006-05-17 EP claimed
WO-2005019216-A1 AMINOBENZIMIDAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2005-03-03 WO claimed