SCHEMBL5809603

SCHEMBL5809603

Fc1ccc(C(F)(F)F)c(C=C2CCN(c3cccnc3)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.43
DPP8 Q6V1X1 2/20 0.43
DPP9 Q86TI2 2/20 0.43
DPP7 Q9UHL4 2/20 0.43
TRPV1 Q8NER1 1/20 0.40
HTR1A P08908 2/20 0.39
DRD4 P21917 2/20 0.39
HTR2A P28223 2/20 0.39
HTR7 P34969 2/20 0.39
DRD3 P35462 2/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
DRD2 P14416 1/20 0.38
CYP11B2 P19099 3/20 0.38
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
CYP19A1 P11511 2/20 0.36
CYP11B1 P15538 2/20 0.36
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5808458 0.78 RBP4 (0.39)
SCHEMBL5805986 0.78 KDM4E (0.44) DPP4DPP8DPP9DPP7HTR1A
SCHEMBL5805823 0.75 PARP1 (0.45)
SCHEMBL5809230 0.75 SLC2A1 (0.44) KDM4E
SCHEMBL5810600 0.72 OGA (0.40) KDM4E
SCHEMBL5806175 0.70 SCD (0.44)
SCHEMBL5806160 0.68 SCD (0.48)
SCHEMBL5810428 0.67 SCD (0.58)
SCHEMBL5808456 0.67 RORC (0.46)
SCHEMBL14824020 0.66 CHRNB2 (0.49) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006125181-A2 PIPERIDINE DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE MODULATORS XENON PHARMACEUTICALS INC. (CA) 2006-11-23 WO disclosed