SCHEMBL5815499

SCHEMBL5815499

CN=C(N)c1c(SC)nc(-c2ccc(SC)cc2)n(-c2ccc(Cl)cc2)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.35
TP53 P04637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
HPGD P15428 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ESR1 P03372 1/20 0.33
CNR1 P21554 1/20 0.32
MAPT P10636 2/20 0.32
HTT P42858 2/20 0.32
AOC3 Q16853 2/20 0.32
PLAU P00749 1/20 0.32
KCNH2 Q12809 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821480 0.92 ALDH1A1 (0.41) ALDH1A1KDM4ENPSR1HPGDRXFP1
SCHEMBL5821418 0.91 TP53 (0.43) PTGS2TP53L3MBTL1ALDH1A1MAPT
SCHEMBL5817548 0.90 DHFR (0.36) ALDH1A1KDM4ERXFP1ESR1MAPT
SCHEMBL5819669 0.88 PTGS2 (0.39) PTGS2ALDH1A1ESR1PLAU
SCHEMBL7245967 0.82 ESR1 (0.39) PTGS2TP53ALDH1A1ESR1MAPT
SCHEMBL5822051 0.81 KATNA1 (0.37) ALDH1A1KDM4EHPGDMAPTHTT
SCHEMBL5821043 0.81 ESR1 (0.35) PTGS2TP53ALDH1A1ESR1CNR1
SCHEMBL5817617 0.80 MAPK14 (0.36) TP53L3MBTL1ALDH1A1NPSR1RXFP1
SCHEMBL4855957 0.78 KDM4E (0.47) PTGS2L3MBTL1ALDH1A1KDM4ENPSR1
SCHEMBL4854626 0.78 KDM4E (0.47) PTGS2L3MBTL1ALDH1A1KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO claimed
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO disclosed