SCHEMBL5819669

SCHEMBL5819669

CN=C(N)c1c(SC)nc(-c2ccc(C(F)(F)F)cc2)n(-c2ccc(SC)cc2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
GABRP O00591 2/20 0.34
GABRD O14764 2/20 0.34
GABRA1 P14867 2/20 0.34
GABRB1 P18505 2/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA5 P31644 2/20 0.34
GABRA3 P34903 2/20 0.34
GABRA2 P47869 2/20 0.34
GABRB2 P47870 2/20 0.34
GABRA4 P48169 2/20 0.34
GABRE P78334 2/20 0.34
GABRA6 Q16445 2/20 0.34
GABRG1 Q8N1C3 2/20 0.34
GABRG3 Q99928 2/20 0.34
GABRQ Q9UN88 2/20 0.34
GRM5 P41594 1/20 0.34
PLAU P00749 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821480 0.90 ALDH1A1 (0.41) PLAUALDH1A1ESR1
SCHEMBL5815499 0.88 PTGS2 (0.35) PTGS2PLAUALDH1A1ESR1
SCHEMBL5817548 0.86 DHFR (0.36) PLAUCYP1A2CYP2C19ALDH1A1ESR1
SCHEMBL5819664 0.82 PTGS2 (0.39) PTGS2PTGS1GABRPGABRDGABRA1
SCHEMBL5817617 0.81 MAPK14 (0.36) SRCKDRALDH1A1MAPK13GCGR
SCHEMBL5822051 0.80 KATNA1 (0.37) PLAUCYP1A2ALDH1A1
SCHEMBL4861654 0.79 PTGS2 (0.42) PTGS2PTGS1GABRPGABRDGABRA1
SCHEMBL5821418 0.78 TP53 (0.43) PTGS2CYP2C19ALDH1A1
SCHEMBL7245244 0.78 MAPK13 (0.40) GABRA2GABRB2ALDH1A1ESR1MAPK13
SCHEMBL5817771 0.76 PTGS2 (0.43) PTGS2PTGS1GRM5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO claimed