SCHEMBL5815501

SCHEMBL5815501

CCOC(=O)N1CCC(c2nc(-c3cccc(Cl)c3)c(-c3ccnc([S+](C)[O-])n3)s2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
MAPT P10636 2/20 0.41
KCNH2 Q12809 2/20 0.40
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
DGAT1 O75907 1/20 0.38
MAPK14 Q16539 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 1/20 0.38
MAP4K4 O95819 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
FNTA P49354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5812539 0.92 NOS3 (0.40) NOS1NOS2MAPTMAPK14KDM4E
SCHEMBL5817168 0.91 MAP4K4 (0.40) KCNH2MAPK14ALDH1A1MAP4K4LMNA
SCHEMBL5814921 0.89 TRPC3 (0.42) MAPTKCNH2MAPK14KDM4EALDH1A1
SCHEMBL5813472 0.86 NOS1 (0.43) NOS1NOS2MAPTKCNH2TP53
SCHEMBL5815240 0.86 MAPK14 (0.49) KCNH2MAPK14
SCHEMBL5817719 0.85 NOS3 (0.41) NOS1NOS2MAPTMAPK14KDM4E
SCHEMBL5815514 0.85 DGAT1 (0.53) NOS1NOS2KCNH2DGAT1MAPK14
SCHEMBL5815323 0.84 DGAT1 (0.52) NOS1NOS2KCNH2DGAT1MAPK14
SCHEMBL5819605 0.83 ALDH1A1 (0.42) NOS2MAPTTP53MAPK14KDM4E
SCHEMBL5818450 0.83 DGAT1 (0.51) NOS1NOS2KCNH2DGAT1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO claimed