SCHEMBL5818904

SCHEMBL5818904

COc1ccc(N2C=Cc3cc(C(C)(C)C)nc(N4CCCCC4)c3C2)cc1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.37
HPGD P15428 5/20 0.37
KDM4E B2RXH2 4/20 0.37
HSD17B10 Q99714 3/20 0.37
ALOX15 P16050 2/20 0.37
USP2 O75604 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TSHR P16473 4/20 0.35
LMNA P02545 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
POLB P06746 2/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821178 0.84 HIF1A (0.39) ALDH1A1HPGDKDM4EHSD17B10ALOX15
SCHEMBL4907061 0.70 EGFR (0.42) ALDH1A1HPGDKDM4EHSD17B10ALOX15
SCHEMBL28860292 0.67 ALDH1A1 (0.63) ALDH1A1HPGDKDM4EALOX15USP2
SCHEMBL5813978 0.65 KDM4E (0.38) ALDH1A1KDM4ETP53MAPK1MAPT
SCHEMBL5815540 0.65 KDM4E (0.42) ALDH1A1KDM4ELMNANPSR1MEN1
SCHEMBL7303075 0.65 ALDH1A1 (0.65) ALDH1A1HPGDKDM4EHSD17B10USP2
SCHEMBL12570448 0.60 MEN1 (0.49) ALDH1A1HPGDKDM4EHSD17B10ALOX15
SCHEMBL2498677 0.58 MEN1 (0.60) ALDH1A1HPGDKDM4EUSP2TDP1
SCHEMBL17241036 0.58 ALDH1A1 (0.54) ALDH1A1KDM4EALOX15USP2TDP1
SCHEMBL20460064 0.57 ALDH1A1 (0.48) ALDH1A1HPGDKDM4EHSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO disclosed