SCHEMBL7303075

SCHEMBL7303075

COc1ccc(N2CCCC2)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.65
LMNA P02545 2/20 0.61
HIF1A Q16665 3/20 0.59
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
NPC1 O15118 1/20 0.56
USP2 O75604 1/20 0.56
RAB9A P51151 1/20 0.56
MAPT P10636 2/20 0.51
KDM4E B2RXH2 2/20 0.51
HPGD P15428 2/20 0.51
POLB P06746 1/20 0.51
HTR7 P34969 1/20 0.50
SLC16A3 O15427 2/20 0.49
SLC16A1 P53985 2/20 0.49
HTT P42858 1/20 0.49
DPP4 P27487 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
CASP1 P29466 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28860292 0.98 ALDH1A1 (0.63) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL2498677 0.85 MEN1 (0.60) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL27988319 0.85 ALDH1A1 (0.49) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL8344083 0.85 ALDH1A1 (0.57) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL13243994 0.85 SIRT6 (0.63) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL12806668 0.85 ALDH1A1 (0.61) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL12856135 0.83 ALDH1A1 (0.59) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL361649 0.83 ADRB1 (0.61) LMNAMAPTHTR7
SCHEMBL15928735 0.83 S100B (0.56) ALDH1A1LMNAHIF1AMEN1KMT2A
SCHEMBL4147257 0.83 ALDH1A1 (0.47) ALDH1A1LMNAHIF1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed
EP-0381235-A2 Pyrrolidine compound and pharmaceutical use Eisai Co., Ltd. (JP) 1990-08-08 EP disclosed