SCHEMBL5821095

SCHEMBL5821095

CNC(=N)c1c(SC)nc(-c2ccc(S(N)(=O)=O)cc2)n(-c2ccc(C)cc2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 10/20 0.43
CA1 P00915 8/20 0.43
CA2 P00918 8/20 0.43
CA12 O43570 7/20 0.43
PTGS2 P35354 8/20 0.42
PTGS1 P23219 3/20 0.42
CA4 P22748 3/20 0.40
ALDH1A1 P00352 1/20 0.40
CHRNA7 P36544 1/20 0.38
CA5A P35218 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820968 0.92 CA2 (0.38) CA9CA1CA2CA12PTGS2
SCHEMBL5817584 0.91 PTGS2 (0.39) CA9CA1CA2CA12PTGS2
SCHEMBL5821476 0.87 ALDH1A1 (0.43) ALDH1A1
SCHEMBL5819681 0.84 CA9 (0.43) CA9CA1CA2CA12PTGS2
SCHEMBL5822322 0.84 CA9 (0.43) CA9CA1CA2CA12PTGS2
SCHEMBL5817785 0.83 ALDH1A1 (0.31) ALDH1A1
SCHEMBL5821043 0.79 ESR1 (0.35) PTGS2ALDH1A1
SCHEMBL6141903 0.79 GAA (0.49) CA9CA1CA2CA12PTGS2
SCHEMBL5815528 0.78 GAA (0.38) CA9CA1CA2CA12PTGS2
SCHEMBL5821416 0.78 AOC3 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129181-A2 PREPARATION OF 4-PYRIMIDONE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2006-12-07 WO claimed