SCHEMBL5828656

SCHEMBL5828656

CC(C)c1c(C(N)=O)ccc(N(c2cc(C(N)=O)ccc2F)C2CCN(Cc3ccncc3)CC2)c1C(C)C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.41
OPRD1 P41143 7/20 0.41
OPRK1 P41145 6/20 0.41
KCNH2 Q12809 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
PARP1 P09874 1/20 0.38
HIF1A Q16665 2/20 0.36
EPAS1 Q99814 2/20 0.36
TLR9 Q9NR96 1/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
IKBKE Q14164 1/20 0.35
TBK1 Q9UHD2 1/20 0.35
GAA P10253 1/20 0.35
ACHE P22303 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5829663 0.90 DRD4 (0.42) OPRM1OPRD1OPRK1KCNH2PARP1
SCHEMBL5829616 0.87 PARP1 (0.40) OPRM1OPRD1OPRK1PARP1GAA
SCHEMBL5829936 0.87 PARP2 (0.40) OPRM1OPRD1OPRK1KCNH2GAA
SCHEMBL5829647 0.86 PARP1 (0.42) OPRM1OPRD1OPRK1PARP1TLR9
SCHEMBL5829864 0.86 PARP1 (0.44) OPRM1OPRD1OPRK1KCNH2HRH3
SCHEMBL5829605 0.85 PARP1 (0.43) OPRM1OPRD1OPRK1KCNH2PARP1
SCHEMBL5828654 0.81 OPRD1 (0.51) OPRM1OPRD1OPRK1KCNH2HRH3
SCHEMBL5630843 0.80 OPRD1 (0.52) OPRM1OPRD1OPRK1
SCHEMBL5879320 0.79 OPRD1 (0.65) OPRM1OPRD1OPRK1
SCHEMBL5629708 0.79 OPRD1 (0.53) OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008952-B2 4-(phenyl-(piperidin-4yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders ASTRAZENECA AB (SE) 2006-03-07 US claimed