SCHEMBL5829616

SCHEMBL5829616

CC(C)c1c(C(N)=O)ccc(N(c2cc(C(N)=O)ccc2F)C2CCN(Cc3ccsc3)CC2)c1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
OPRM1 P35372 10/20 0.39
OPRD1 P41143 8/20 0.39
ARRB1 P49407 1/20 0.38
OPRK1 P41145 7/20 0.38
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
F10 P00742 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
GAA P10253 1/20 0.32
TNIK Q9UKE5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6613888 0.87 OPRM1 (0.49) PARP1PARP2OPRM1OPRD1ARRB1
SCHEMBL5828656 0.87 OPRM1 (0.41) PARP1OPRM1OPRD1OPRK1GAA
SCHEMBL6751101 0.86 PARP1 (0.46) PARP1PARP2OPRM1OPRD1ARRB1
SCHEMBL5829605 0.85 PARP1 (0.43) PARP1PARP2OPRM1OPRD1OPRK1
SCHEMBL5829936 0.85 PARP2 (0.40) PARP2OPRM1OPRD1OPRK1CHRM2
SCHEMBL5829663 0.84 DRD4 (0.42) PARP1PARP2OPRM1OPRD1OPRK1
SCHEMBL5829612 0.82 OPRD1 (0.48) OPRM1OPRD1ARRB1OPRK1
SCHEMBL5829647 0.82 PARP1 (0.42) PARP1OPRM1OPRD1OPRK1ALDH1A1
SCHEMBL5879344 0.80 OPRD1 (0.60) OPRM1OPRD1OPRK1
SCHEMBL5630843 0.77 OPRD1 (0.52) OPRM1OPRD1OPRK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008952-B2 4-(phenyl-(piperidin-4yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders ASTRAZENECA AB (SE) 2006-03-07 US claimed