SCHEMBL5829936

SCHEMBL5829936

CC(C)c1c(C(N)=O)ccc(N(c2cc(C(N)=O)ccc2F)C2CCN(Cc3ccoc3)CC2)c1C(C)C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP2 Q9UGN5 1/20 0.40
OPRM1 P35372 8/20 0.39
OPRD1 P41143 8/20 0.39
OPRK1 P41145 7/20 0.38
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
HRH2 P25021 1/20 0.34
CACNA2D1 P54289 1/20 0.33
CHRM4 P08173 1/20 0.32
SSTR5 P35346 1/20 0.32
KCNH2 Q12809 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
MCHR1 Q99705 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828656 0.87 OPRM1 (0.41) OPRM1OPRD1OPRK1KCNH2GAA
SCHEMBL5830029 0.86 PARP2 (0.46) PARP2OPRM1OPRD1OPRK1HTR2A
SCHEMBL5829616 0.85 PARP1 (0.40) PARP2OPRM1OPRD1OPRK1CHRM2
SCHEMBL5829663 0.84 DRD4 (0.42) PARP2OPRM1OPRD1OPRK1KCNH2
SCHEMBL5829605 0.84 PARP1 (0.43) PARP2OPRM1OPRD1OPRK1HRH2
SCHEMBL5829932 0.82 OPRD1 (0.48) OPRM1OPRD1OPRK1
SCHEMBL5829647 0.82 PARP1 (0.42) OPRM1OPRD1OPRK1
SCHEMBL5879372 0.80 OPRD1 (0.60) OPRM1OPRD1OPRK1
SCHEMBL5630843 0.77 OPRD1 (0.52) OPRM1OPRD1OPRK1
SCHEMBL5629708 0.76 OPRD1 (0.53) OPRM1OPRD1OPRK1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7008952-B2 4-(phenyl-(piperidin-4yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders ASTRAZENECA AB (SE) 2006-03-07 US claimed