SCHEMBL5828878

SCHEMBL5828878

COc1cc2ncnc(N/C(=N\CCC3CCCN3C)Nc3c(C)cccc3C)c2cc1OC

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.51
EPHA2 P29317 1/20 0.51
EPHB4 P54760 1/20 0.51
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
EGFR P00533 7/20 0.42
NSD2 O96028 1/20 0.42
ERBB2 P04626 1/20 0.41
RET P07949 5/20 0.41
KIF5B P33176 5/20 0.41
FGFR1 P11362 2/20 0.41
FLT1 P17948 2/20 0.41
CDK2 P24941 1/20 0.41
PIK3R1 P27986 1/20 0.41
EPHB2 P29323 1/20 0.41
TTBK1 Q5TCY1 1/20 0.41
NOD1 Q9Y239 1/20 0.40
AURKA O14965 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828880 1.00 KDR (0.51) KDREPHA2EPHB4ALDH1A1HPGD
SCHEMBL5828980 0.94 KDR (0.46) KDREPHA2EPHB4EGFRRET
SCHEMBL5828988 0.94 KDR (0.46) KDREPHA2EPHB4EGFRRET
SCHEMBL5828058 0.94 KDR (0.48) KDREPHA2EPHB4HPGDHTT
SCHEMBL5828053 0.94 KDR (0.48) KDREPHA2EPHB4HPGDHTT
SCHEMBL6981911 0.80 HTT (0.48) KDRALDH1A1HPGDHTTEGFR
SCHEMBL6985649 0.78 RET (0.49) KDRALDH1A1HPGDHTTEGFR
SCHEMBL7089596 0.78 KDR (0.48) KDREPHA2EPHB4HPGDHTT
SCHEMBL7090020 0.78 KDR (0.45) KDREPHA2EPHB4EGFRRET
SCHEMBL6980090 0.77 EGFR (0.60) KDREGFRRETKIF5BFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7001904-B1 Guanidine derivatives quinazoline and quinoline for use in the treatment of autoimmune diseases ASTRAZENECA AB (SE) 2006-02-21 US disclosed