SCHEMBL5830288

SCHEMBL5830288

C=C(C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1)c1ccc(Sc2ccccc2Br)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 12/20 0.49
CHRM1 P11229 2/20 0.49
PLD2 O14939 2/20 0.48
PLD1 Q13393 2/20 0.48
AVPR1A P37288 2/20 0.46
HTR1A P08908 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
TACR2 P21452 1/20 0.45
DRD1 P21728 1/20 0.45
DRD5 P21918 1/20 0.45
SLC6A2 P23975 1/20 0.45
ADRA1D P25100 1/20 0.45
HTR1B P28222 1/20 0.45
TSPO P30536 1/20 0.45
ADORA1 P30542 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6197862 0.82 PDE7A (0.41) ALDH1A1
SCHEMBL6310726 0.81 ITGB2 (0.50) HSD11B1CHRM1AVPR1AHTR1AADORA3
SCHEMBL5830031 0.79 PDE7A (0.44) HSD11B1ALDH1A1
SCHEMBL7702269 0.77 ITGB2 (0.48) ALDH1A1
SCHEMBL5830183 0.76 PDE7A (0.36) ALDH1A1
SCHEMBL5836083 0.75 ITGAL (0.41) ALDH1A1MAPK1
SCHEMBL5829934 0.73 EPHX2 (0.40) CHRM1ALDH1A1
SCHEMBL5830812 0.73 SPR (0.42) ALDH1A1
SCHEMBL6494066 0.72 AKR1C3 (0.40) ALDH1A1
SCHEMBL6494059 0.72 PDE7A (0.36) HSD11B1TACR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39197-E1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2006-07-18 US claimed
EP-1140814-B1 CELL ADHESION-INHIBITING ANTIINFLAMMATORY AND IMMUNE-SUPPRESSIVE COMPOUNDS ABBOTT LAB (US) 2005-05-25 EP claimed
US-6878700-B1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2005-04-12 US claimed
US-6878700-B1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2005-04-12 US disclosed
US-6867203-B2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2005-03-15 US disclosed
US-20040116518-A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES 2004-06-17 US disclosed