SCHEMBL5837565

SCHEMBL5837565

Cc1cc2c(c(Sc3ccc(Cl)cc3)n1)C(=O)N(CC1Cc3c(sc(NC(=O)C(=O)OC(C)(C)C)c3C(=O)OC(C)(C)C)CO1)C2=O

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.33
ALDH1A1 P00352 2/20 0.31
TSHR P16473 1/20 0.31
CXCR2 P25025 3/20 0.31
MAPT P10636 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5839221 0.89 ADORA1 (0.36) GPR119
SCHEMBL5838631 0.87 PTPN1 (0.37) GPR119ALDH1A1TSHR
SCHEMBL5838083 0.81 CXCR2 (0.31) CXCR2
SCHEMBL5846957 0.80 GPR119 (0.33) GPR119ALDH1A1TSHR
SCHEMBL5837378 0.78 ALDH1A1 (0.44) ALDH1A1TSHR
SCHEMBL5838538 0.77 CXCR2 (0.37) ALDH1A1TSHRCXCR2MAPT
SCHEMBL5838589 0.77 CXCR2 (0.37) ALDH1A1TSHRCXCR2MAPTRXFP1
SCHEMBL5837569 0.71 CXCR2 (0.42) ALDH1A1CXCR2MAPT
SCHEMBL5838393 0.70 CXCR2 (0.41) ALDH1A1CXCR2MAPT
SCHEMBL5839226 0.69 ADORA1 (0.35) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115624-B1 Method of inhibiting protein tyrosine phosphatase 1B and/or T-cell protein tyrosine phosphatase 4 and/or other PTPases with an Asp residue at position 48 NOVO NORDISK A/S (DK) 2006-10-03 US disclosed