SCHEMBL5838696

SCHEMBL5838696

CC(C)(C)OC(=O)c1c(CN2C(=O)c3cccc([N+](=O)[O-])c3C2=O)sc2c1CCOC2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 6/20 0.42
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 4/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MAPT P10636 2/20 0.38
ATM Q13315 1/20 0.37
LMNA P02545 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571114 0.78 CXCR2 (0.46) CXCR2MAPTACHE
SCHEMBL5838706 0.76 CXCR2 (0.42) CXCR2
SCHEMBL5838657 0.75 ALDH1A1 (0.37) TDP1ALDH1A1CA12CA1CA2
SCHEMBL5838700 0.71 TDP1 (0.39) TDP1ALDH1A1CA12CA1CA2
SCHEMBL14876479 0.70 ATM (0.56) TDP1ALDH1A1CA12CA1CA2
SCHEMBL26744283 0.68 ALDH1A1 (0.53) TDP1ALDH1A1CA12CA1CA2
SCHEMBL30050782 0.65 CA1 (0.59) TDP1ALDH1A1CA12CA1CA2
SCHEMBL4375792 0.65 CA1 (0.59) TDP1ALDH1A1CA12CA1CA2
SCHEMBL6315716 0.64 CXCR2 (0.54) CXCR2ALDH1A1MAPTLMNA
SCHEMBL5838665 0.62 ADORA1 (0.33) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115624-B1 Method of inhibiting protein tyrosine phosphatase 1B and/or T-cell protein tyrosine phosphatase 4 and/or other PTPases with an Asp residue at position 48 NOVO NORDISK A/S (DK) 2006-10-03 US disclosed