SCHEMBL5839465

SCHEMBL5839465

O=C(O)c1ccccc1OCc1cccc(OC(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 7/20 0.56
RXRA P19793 1/20 0.52
RXRB P28702 1/20 0.52
RXRG P48443 1/20 0.52
KDM5A P29375 1/20 0.50
KDM4C Q9H3R0 1/20 0.50
KDM5B Q9UGL1 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPK14 Q16539 1/20 0.48
CTSV O60911 1/20 0.48
CTSL P07711 1/20 0.48
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP14 P50281 1/20 0.47
ADAM17 P78536 1/20 0.47
USP28 Q96RU2 1/20 0.47
USP25 Q9UHP3 1/20 0.47
PTGER1 P34995 1/20 0.47
FOLH1 Q04609 1/20 0.47
FFAR1 O14842 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2447727 0.85 RXRA (0.63) MRGPRX4RXRARXRBRXRGALDH1A1
SCHEMBL5839266 0.84 FFAR1 (0.56) MRGPRX4ALDH1A1CTSVCTSLPTGER1
SCHEMBL1388008 0.83 MRGPRX4 (0.59) MRGPRX4ALDH1A1PTGER1
SCHEMBL2453780 0.82 NR4A2 (0.62) MRGPRX4ALDH1A1FFAR1NR4A2
SCHEMBL27436417 0.81 MRGPRX4 (0.53) MRGPRX4RXRARXRBRXRGKDM5A
SCHEMBL3375496 0.80 MRGPRX4 (0.62) MRGPRX4MAPK14MMP2MMP9MMP14
SCHEMBL9138058 0.80 KDM4E (0.51) KDM5AKDM4CKDM5BALDH1A1MAPK14
SCHEMBL2453382 0.80 LMNA (0.62) MRGPRX4ALDH1A1PTGER1FOLH1NR4A2
SCHEMBL12189462 0.79 MRGPRX4 (0.53) MRGPRX4
SCHEMBL112903 0.79 SGMS2 (0.66) ALDH1A1PTGER1FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6984645-B2 Dual inhibitors of adipocyte fatty acid binding protein and keratinocyte fatty acid binding protein BRISTOL-MYERS SQUIBB COMPANY (US) 2006-01-10 US disclosed