SCHEMBL5845974

SCHEMBL5845974

O=C(O)CNC(=O)OCCNc1nc2ccccc2[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.57
ALPL P05186 2/20 0.49
ALPG P10696 2/20 0.49
PLAA Q9Y263 1/20 0.49
TRPC3 Q13507 1/20 0.49
TRPC4 Q9UBN4 1/20 0.49
TRPC5 Q9UL62 1/20 0.49
KCNH2 Q12809 2/20 0.48
RAB9A P51151 5/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
TP53 P04637 2/20 0.48
NPC1 O15118 4/20 0.46
ALDH1A1 P00352 2/20 0.46
ALOX12 P18054 1/20 0.46
HSD17B10 Q99714 2/20 0.46
MAPK1 P28482 1/20 0.46
PKM P14618 1/20 0.46
MAOB P27338 1/20 0.46
ADORA2A P29274 1/20 0.46
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5845732 0.81 BCHE (0.60) BCHEALPLALPGPLAATRPC3
SCHEMBL5844227 0.81 ITGB3 (0.47) BCHEALPLALPGPLAARAB9A
SCHEMBL8328333 0.80 ALPL (0.64) BCHEALPLALPGPLAATRPC3
SCHEMBL5846138 0.80 KCNH2 (0.60) BCHEALPLALPGPLAATRPC3
SCHEMBL7217435 0.78 BCHE (0.60) BCHEALPLALPGPLAATRPC3
SCHEMBL16866616 0.77 BCHE (0.55) BCHEALPLALPGPLAATRPC3
SCHEMBL6764617 0.76 BCHE (0.65) BCHEALPLALPGPLAATRPC3
SCHEMBL13049808 0.74 BCHE (0.66) BCHETRPC3TRPC4TRPC5KCNH2
SCHEMBL17329389 0.73 BCHE (0.57) BCHEALPLALPGPLAATRPC3
SCHEMBL5844930 0.72 BCHE (0.67) BCHEALPLALPGPLAATRPC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7135587-B2 Urea and urethane derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2006-11-14 US disclosed
EP-1343764-B1 UREA AND URETHANE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2004-08-25 EP disclosed
US-20040063644-A1 Urea and urethane derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063644-A1 Urea and urethane derivatives as integrin inhibitors ITGB1, ITGB2, ITGA1 BCHE 3836/4885ALPL 3246/4885ALPG 3535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.