SCHEMBL5847121

SCHEMBL5847121

COc1ccc(-c2cc3c4c(c2C(C)(C)C)[C@@H]2CN(C(=O)O)CC[C@@H]2N4CC3)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 2/20 0.35
MCHR1 Q99705 5/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
FFAR1 O14842 1/20 0.33
ESR1 P03372 2/20 0.32
ESR2 Q92731 1/20 0.32
ALDH1A1 P00352 4/20 0.32
HSD11B1 P28845 1/20 0.31
RORC P51449 1/20 0.31
MTNR1B P49286 1/20 0.31
NOTUM Q6P988 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847619 0.90 CPS1 (0.37) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5847193 0.90 CCR3 (0.35) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5847324 0.90 CCR3 (0.34) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5847800 0.89 HTR2A (0.44) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5846973 0.89 CCR3 (0.34) CCR3MCHR1HTR2AHTR2CHTR2B
SCHEMBL5849715 0.87 DRD1 (0.37) CCR3HTR2AHTR2C
SCHEMBL5849356 0.84 CCR3 (0.30) CCR3
SCHEMBL5847913 0.82 ABCB1 (0.35) CCR3HTR2CALDH1A1
SCHEMBL5847854 0.82 HCRTR1 (0.36) CCR3HTR2AHTR2C
SCHEMBL5410492 0.81 HTR2C (0.46) CCR3MCHR1HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed