SCHEMBL5846973

SCHEMBL5846973

COc1ccc(-c2cc3c4c(c2C(C)(C)C)[C@@H]2CN(C(=O)O)CC[C@@H]2N4CC3)c(C(C)C)c1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
ABCB1 P08183 2/20 0.32
POLB P06746 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
ABHD6 Q9BV23 1/20 0.31
MCHR1 Q99705 1/20 0.31
DPP4 P27487 1/20 0.30
DPP7 Q9UHL4 1/20 0.30
HPGD P15428 1/20 0.30
MGLL Q99685 1/20 0.30
RORC P51449 1/20 0.30
FKBP1A P62942 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847121 0.89 CCR3 (0.35) CCR3HTR2AHTR2CHTR2BMTNR1B
SCHEMBL5847193 0.88 CCR3 (0.35) CCR3HTR2AHTR2CHTR2BMTNR1A
SCHEMBL5847619 0.88 CPS1 (0.37) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5847324 0.87 CCR3 (0.34) CCR3HTR2AHTR2CHTR2BMTNR1B
SCHEMBL5847800 0.87 HTR2A (0.44) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5416032 0.82 HTR2C (0.44) CCR3HTR2AHTR2CHTR2BMTNR1A
SCHEMBL5847913 0.82 ABCB1 (0.35) CCR3HTR2CABCB1POLBHPGD
SCHEMBL5847475 0.82 S1PR1 (0.37) HTR2AHTR2CHTR2BDPP4
SCHEMBL5847854 0.80 HCRTR1 (0.36) CCR3HTR2AHTR2CDPP4DPP7
SCHEMBL5847306 0.80 HTR2A (0.36) HTR2AHTR2CHTR2BMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed