SCHEMBL5847619

SCHEMBL5847619

COc1ccc(-c2cc3c4c(c2C(C)(C)C)[C@@H]2CN(C(=O)O)CC[C@@H]2N4CC3)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CPS1 P31327 14/20 0.37
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
RORC P51449 1/20 0.35
CCR3 P51677 2/20 0.35
JAK2 O60674 1/20 0.34
JAK3 P52333 1/20 0.34
PTK2 Q05397 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847121 0.90 CCR3 (0.35) HTR2AHTR2CHTR2BRORCCCR3
SCHEMBL5847800 0.90 HTR2A (0.44) HTR2AHTR2CHTR2BCCR3ESR1
SCHEMBL5847193 0.90 CCR3 (0.35) HTR2AHTR2CHTR2BCCR3ESR1
SCHEMBL5847324 0.89 CCR3 (0.34) HTR2AHTR2CHTR2BRORCCCR3
SCHEMBL5846973 0.88 CCR3 (0.34) HTR2AHTR2CHTR2BRORCCCR3
SCHEMBL5848064 0.88 DPP4 (0.36) CCR3
SCHEMBL5849356 0.84 CCR3 (0.30) CCR3
SCHEMBL5847913 0.82 ABCB1 (0.35) HTR2CCCR3
SCHEMBL5847475 0.82 S1PR1 (0.37) HTR2AHTR2CHTR2B
SCHEMBL5847854 0.82 HCRTR1 (0.36) HTR2AHTR2CCCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed